产品
编 号:F741706
分子式:C19H18N6S
分子量:362.45
产品类型
结构图
CAS No: 2649882-80-2
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产品详情
生物活性:
ARN25068 is a sub-micromolar inhibitor of the three protein kinases, GSK-3β, FYN and DYRK1A to tackle tau hyperphosphorylation.
体外研究:
ARN25068 reduces the extent of tau phosphorylation in Tau0N4R-TM-tGFP U2OS cell line. ARN25068 exhibits IC50 values of 4.17 and 2.17 μM for GSK-3β and FYN in enzymatic radiometric assay, respectively.