产品
编 号:F741661
分子式:C30H34F3N5O
分子量:537.62
产品类型
结构图
CAS No: 2573775-59-2
联系客服
产品详情
生物活性:
Cbl-b-IN-3 (Compound 23) is a casitas B-lineage lymphoma proto-oncogene-b (Cbl-b) inhibitor with an IC50 of < 1 nM. Cbl-b is an E3 ubiquitin ligase that negatively regulates T-cell activation.
体外研究:
Cbl-b-IN-3 (Compound 23) enhances IL-2 secretion by T-cells stimulated with an anti-CD3 antibody alone or in combination with an anti-CD28 antibody.