产品
编 号:F727351
分子式:C24H23NO2
分子量:357.44
产品类型
结构图
CAS No: 1141802-49-4
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产品详情
生物活性:
LUF5771 is a potent allosteric recombinant luteinizing hormone (recLH) and Org 43553 inhibitor. LUF5771 is able to partially activate the LH receptor with low efficacy.
体外研究:
LUF5771 (1 μM or 10 μM) allosteric inhibition is concentration-dependent. LUF5771 significantly increases radioligand dissociation. LUF5771 probably binds to the seven transmembrane domain like Org 43553 does. LUF5771 (10 μM) alone is able to partially activate the LH receptor by 31±4%.