产品
编 号：F717605
分子式：C29H43NO3
分子量：453.66
分子式：C29H43NO3
分子量：453.66
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CAS No: 616884-65-2
产品详情
生物活性：
OMDM-4 is a selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki 17.7 μM.
体外研究：
OMDM-4 shows poor affinity for either CB1 (Ki=4.9 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively. OMDM-4 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50>10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM).
OMDM-4 is a selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki 17.7 μM.
体外研究：
OMDM-4 shows poor affinity for either CB1 (Ki=4.9 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively. OMDM-4 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50>10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM).
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