产品
编 号:F701518
分子式:C29H36N4O3
分子量:488.62
产品类型
结构图
CAS No: 1638526-94-9
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产品详情
生物活性:
Bax activator-1 (compound 106) is a Bax activator that induces Bax-dependent tumor cell apoptosis.
体内研究:
Bax activator-1 (40 mg/kg; given i.p., each day for 13 days) inhibits lung tumor growth in C57BL/6 female mice.Animal Model:Eight-week old C57BL/6 female mice (with Lewis Lung Carcinoma tumor cells)
Dosage:40 mg/kg
Administration:Given i.p., each day for 13 days
Result:Exhibited anti-tumor activity as a single-agent.
体外研究:
Bax activator-1 (20-80 μM; 48 hours) induces Bax-dependent tumor cell apoptosis in a dose-dependent fashion.