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编 号:F700083
分子式:C25H28ClF3N4O4
分子量:540.96
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BMS-986118 is a potent, orally active, and selective GPR40 agonist with an EC50 of 0.07 μM. BMS-986118 has dual insulinotropic and GLP-1 secretory effects, resulting in robust plasma glucose lowering effects in acute animal models.
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