产品
编 号：F673596
分子式：C24H33ClN2O3
分子量：432.98
分子式：C24H33ClN2O3
分子量：432.98
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CAS No: 124439-07-2
产品详情
生物活性：
Enadoline (CI-977) hydrochloride is a highly selective, brain-penetrating, and nonpeptide kappa-opioid receptor (KOR) agonist (Ki=1.25 nM). Antinociceptive effects.
体内研究：
Enadoline (i.v.; dose of e 15 min before surgery; male Sprague-Dawley rats) hydrochloride dose-dependently (1-100 μg/kg) blocks the development of thermal hyperalgesia as well as static and dynamic allodynia for over 24 h with respective MEDs (minimum effective doses) of < or = 1, 10 and 10 μg/kg.
Enadoline (CI-977) hydrochloride is a highly selective, brain-penetrating, and nonpeptide kappa-opioid receptor (KOR) agonist (Ki=1.25 nM). Antinociceptive effects.
体内研究：
Enadoline (i.v.; dose of e 15 min before surgery; male Sprague-Dawley rats) hydrochloride dose-dependently (1-100 μg/kg) blocks the development of thermal hyperalgesia as well as static and dynamic allodynia for over 24 h with respective MEDs (minimum effective doses) of < or = 1, 10 and 10 μg/kg.
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