产品
编 号:F672322
分子式:C22H25NO5S
分子量:415.5
产品类型
结构图
CAS No: 1228439-71-1
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产品详情
生物活性:
(+)-KCC2 blocker 1 is a selective K+-Cl- cotransporter KCC2 blocker with an IC50 of 0.4 μM. (+)-KCC2 blocker 1 is a benzyl prolinate and a enantiomer of KCC2 blocker 1.
体外研究:
(+)-KCC2 blocker 1 ((+)-13), a enantiomers of KCC2 blocker 1, has a 100-fold difference in potency compare with enantiomer (-)-KCC2 blocker 1 ((?)-13)).