产品
编 号:F667827
分子式:C22H35NO2
分子量:345.52
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5mg
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生物活性:
LY255582 is a pan-opioid antagonist and has high affinity for mu, delta, and kappa receptors (Ki: 0.4 nM, 5.2, 2.0 nM respectively). LY255582 can decrease food intake and body weight. LY255582 can be used for the research of obesity.

体内研究:
LY255582 (100 μg,i.c.v.) 减少大鼠的食物摄入量。LY255582 (15 mg/kg,皮下注射,每日一次) 减少喂食的肥胖 Zucker 大鼠的食物摄入量和体重增加。Animal Model:STZ-induced diabetic mice
Dosage:100, 10 and 1 μg
Administration:i.c.v.
Result:Decreased food at 100, 10 and 1 μg by 76, 62 and 29%.

体外研究:
LY255582 (40 μM, 24-72 h) 抑制 Huh7 和 MHCC-97H 细胞活力。
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