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编 号:F625869
分子式:C12H22F6N4O5
分子量:416.32
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生物活性:
hDDAH-1-IN-1 TFA (compound 8a) is a potent and selective non-amino acid catalytic site inhibitor of human dimethylarginine dimethylaminohydrolase-1 (hDDAH-1), with a Ki of 18 μM.

体外研究:
hDDAH-1-IN-1 TFA potently inhibits hDDAH-1 (Ki = 18 μM) without significantly affecting NOSs and arginase.
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