产品
编 号:F622682
分子式:C36H38BrN3O6
分子量:688.61
产品类型
结构图
CAS No: 1592908-16-1
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产品详情
生物活性:
MSN-125 is a potent Bax and Bak oligomerization inhibitor. MSN-125 prevents mitochondrial outer membrane permeabilization (MOMP) with an IC50 of 4 μM. MSN-125 potently inhibits Bax/Bak-mediated apoptosis in HCT-116, BMK Cells, and primary cortical neurons, protects primary neurons against glutamate excitotoxicity.
体外研究:
MSN-125 以浓度依赖性方式抑制 tBid/Bax 介导的 MOMP。