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编 号:F622368
分子式:C24H27Cl2N7
分子量:484.42
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生物活性:
EAD1 is a potent autophagy inhibitor with antiproliferative activity in lung and pancreatic cancer cells. EAD1 also induces apoptosis.

体外研究:
EAD1 (0-200 μM; 72 hours) has antiproliferative activity against human cancer cell lines.EAD1 (5-75 μM; 24 hours) induces apoptosis in the H460 cells in a concentration-dependent manner. EAD1 (1-25 μM; 24 hour) increases the punctate LC3 signal in H460 cells.
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