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编 号:F522852
分子式:C12H10N6O
分子量:254.25
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10mM*1mL in DMSO
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1mg
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5mg
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10mg
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50mg
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生物活性:
TG 100713 is an inhibitor of PI3K, with IC50s of 24, 50, 165, and 215 nM for PI3Kδ, γ, α and β isoforms respectively.

体外研究:
TG100713 (10 μM; 48 or 72 h) strongly inhibits endothelial cell (EC) proliferation.
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