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编 号:F522828
分子式:C18H14FN5O
分子量:335.34
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10mM*1mL in DMSO
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5mg
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10mg
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25mg
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生物活性:
LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist.

体内研究:
At 3 mg/kg, LAS101057 is active in preventing Acetyl-β-methylcholine-induced AHR, and at 10 mg/kg it inhibits AHR to Acetyl-β-methylcholine to a level virtually equal to that seen with Hexadecadrol at 1 mg/kg.
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