产品
编 号:F520449
分子式:C24H23Cl2N3O
分子量:440.36
产品类型
结构图
CAS No: 919077-81-9
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产品详情
生物活性:
CB2 receptor agonist 3 is a robust and selective CB2 cannabinoid agonist with Kis of 7.6 and 900 nM for CB2 and CB1, respectively. CB2 receptor agonist 3 significantly increases P-ERK 1/2 expression in HL-60 cells.
体外研究:
CB2 receptor agonist 3 (Compound 2a) is also shown to be agonist in an in vitro model based on human promyelocytic leukemia HL-60 cells.