产品
编 号:F511253
分子式:C19H19ClFN5O3
分子量:419.84
产品类型
结构图
CAS No: 900510-03-4
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生物活性:
Cligosiban (PF-3274167), a high oral bioavailability and good brain-penetrant non-peptide oxytocin receptor antagonist, shows a high-affinity (Ki=9.5 nM) and an excellent selectivity versus the vasopressin receptors with almost no affinity for the V1b and V1a subtypes. Cligosiban inhibits ejaculatory physiology in rodents.