产品
编 号:F477705
分子式:C21H22ClFN4O3
分子量:432.88
产品类型
结构图
CAS No: 847949-49-9
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生物活性:
O-Desmethyl gefitinib is an active metabolite of Gefitinib in human plasma. The formation of O-desmethyl gefitinib is dependent on CYP2D6 activity. O-desmethyl gefitinib inhibits EGFR with an IC50 of 36 nM in subcellular assays.