产品
编 号:F476086
分子式:C13H15N3O2S
分子量:277.34
产品类型
结构图
CAS No: 84468-24-6
联系客服
产品详情
生物活性:
HA-100 is a potent protein kinase inhibitor, with IC50s of 4 μM, 8 μM, 12 μM and 240 μM for cGMP-dependent protein kinase (PKG), cAMP-dependent protein kinase (PKA), protein kinase C (PKC) and MLC-kinase, respectively. HA-100 also used as a ROCK inhibitor.
体外研究:
HA-100对mlc -激酶和PKC的ATP具有竞争性抑制作用,Kis分别为 61 μM 和 6.5 μM。