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编 号:F473402
分子式:C21H15ClF4N4O4
分子量:498.81
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10mM*1mL in DMSO
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1mg
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5mg
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10mg
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生物活性:
Regorafénib N-oxyde M2 is an active metabolite of Regorafenib. Regorafenib is a multi-target inhibitor for VEGFR1/2/3, PDGFRβ, Kit, RET and Raf-1 with IC50s of 13/4.2/46, 22, 7, 1.5 and 2.5 nM, respectively.
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