产品
编 号：F472893
分子式：C29H37N5O5
分子量：535.63
分子式：C29H37N5O5
分子量：535.63
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CAS No: 83397-56-2
产品详情
生物活性：
PL-017 is a potent and selective μ opioid receptor agonist with an IC50 of 5.5 nM for 125I-FK 33,824 binding to μ site. PL-017 produces long-lasting, reversible analgesia in rats.
体内研究：
PL-017 (0.22, 0.45, 0.9 nmol/rat; i.c.v.) has the time of maximum effect of approximately 15 to 30 mm after injection at lower doses and produces analgesia lasting as long as 4 hours with larger doses in male Sprague-Dawley rats weighing 250 to 375 g.
体外研究：
PL-017 has an IC50 of 10000 nM for 125I-DADLE binding to δ site.
PL-017 is a potent and selective μ opioid receptor agonist with an IC50 of 5.5 nM for 125I-FK 33,824 binding to μ site. PL-017 produces long-lasting, reversible analgesia in rats.
体内研究：
PL-017 (0.22, 0.45, 0.9 nmol/rat; i.c.v.) has the time of maximum effect of approximately 15 to 30 mm after injection at lower doses and produces analgesia lasting as long as 4 hours with larger doses in male Sprague-Dawley rats weighing 250 to 375 g.
体外研究：
PL-017 has an IC50 of 10000 nM for 125I-DADLE binding to δ site.
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