产品
编 号:F401241
分子式:C21H22ClFN4O2
分子量:416.88
产品类型
结构图
CAS No: 59831-65-1
联系客服
产品详情
生物活性:
Halopemide is a potent phospholipase D (PLD) inhibitor, with IC50s of 220 and 310 nM for human PLD1 and PLD2, respectively. Halopemid is a dopamine receptors antagonist, and acts a psychotropic agent.
体内研究:
Halopemide (10 mg/kg; p.o.) induces dyskinesias in the majority of monkeys tested.
体外研究:
Halopemide (1-2 μM; 21 day) affects calcification in transdifferentiated MOVAS cells.