产品
编 号:F044043
分子式:C8H13N6O4P
分子量:288.2
产品类型
结构图
CAS No: 113852-41-8
联系客服
产品详情
生物活性:
PMEDAP is a potent inhibitor of human immunodeficiency virus (HIV) replication. PMEDAP has anti-murine cytomegalovirus (MCMV) activity. PMEDAP is a very potent inhibitor of Moloney murine sarcoma virus (MSV)-induced tumor formation and associated mortality.
体内研究:
PMEDAP (0.25-5 mg/kg; IP; daily; starting on the day of MSV-infected and continuing for an additional four days) causes a dose-dependent suppression of tumor formation and mortality in newborn mice inoculated with MSV.Animal Model:Three-week-old male NMRI mice
Dosage:0.25 mg/kg, 1 mg/kg, 5 mg/kg
Administration:IP; daily; starting on the day of infection and continuing for an additional four days
Result:Effected a significant delay in tumor appearance and an enhancement of the survival rate of tumor-bearing mice.