产品
编 号:F381304
分子式:C10H8O3
分子量:176.17
产品类型
结构图
CAS No: 531-59-9
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产品详情
生物活性:
Herniarin is a natural coumarin occurs in some flowering plants, with antitumor effect.
体外研究:
Herniarin is cytotoxic to breast carcinoma cell line MCF-7 with an IC50 of 207.6 μM. Herniarin (100 μM) also induces apoptosis in MCF-7 cells. Herniarin alone has no obvious cytotoxicity on transitional cell carcinoma (TCC) cells, but when in combination with 5?μg/mL cisplatin, Herniarin (80 μg/mL) potently enhances the antitumor effect of cisplatin, and increases chromatin condensation.