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编 号:F367771
分子式:C11H14N2O
分子量:190.24
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10mM*1mL in DMSO
询价
询价
5mg
160
In-stock
10mg
240
In-stock
25mg
320
In-stock
50mg
416
In-stock
100mg
544
In-stock
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生物活性:
Cytisinicline (Cytisine) is an alkaloid. Cytisinicline (Cytisine) is a partial agonist of α4β2 nAChRs, and partial to full agonist at β4 containing receptors and α7 receptors. Has been used medically to help with smoking cessation.

体内研究:
Cytisinicline (Cytisine) (5 mg/kg,ip) 比接受载体的那些吃得更少,体重增加也更少。与尼古丁相比,Cytisinicline (Cytisine) 替代期间,总颗粒摄入量增加,而动物自用 Cytisine 明显少于尼古丁。

体外研究:
Cytisinicline (Cytisine) (2.5、5 和 10 mM) 能够诱导 HepG2 细胞凋亡。 G1期 (PCytisinicline 相关抗体:
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