产品
编 号:F367771
分子式:C11H14N2O
分子量:190.24
产品类型
结构图
CAS No: 485-35-8
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产品详情
生物活性:
Cytisinicline (Cytisine) is an alkaloid. Cytisinicline (Cytisine) is a partial agonist of α4β2 nAChRs, and partial to full agonist at β4 containing receptors and α7 receptors. Has been used medically to help with smoking cessation.
体内研究:
Cytisinicline (Cytisine) (5 mg/kg,ip) 比接受载体的那些吃得更少,体重增加也更少。与尼古丁相比,Cytisinicline (Cytisine) 替代期间,总颗粒摄入量增加,而动物自用 Cytisine 明显少于尼古丁。
体外研究:
Cytisinicline (Cytisine) (2.5、5 和 10 mM) 能够诱导 HepG2 细胞凋亡。 G1期 (PCytisinicline 相关抗体: