产品
编 号：F358237
分子式：C11H6F3NO2S
分子量：273.23
分子式：C11H6F3NO2S
分子量：273.23
产品类型
规格
价格
是否有货
5mg
询价
询价
10mg
询价
询价
25mg
询价
询价
50mg
询价
询价
100mg
询价
询价
结构图
CAS No: 438190-29-5
产品详情
生物活性：
SMI-4a (TCS-PIM-1-4a) is a poten, selective, cell-permeable and ATP-competitive Pim-1 inhibitor with an IC50 of 24 μM and a Ki of 0.6 μM. SMI-4a also inhibits Pim-2 (IC50 of 100 μM), and does not significantly inhibit the other serine/threonine- or tyrosine-kinases. SMI-4a has anticancer activity.
体外研究：
SMI-4a (0.5 μM；1 小时；HEK-293T 细胞) 处理会减弱完整细胞中标记的 Pim-1 的自身磷酸化。
SMI-4a (TCS-PIM-1-4a) is a poten, selective, cell-permeable and ATP-competitive Pim-1 inhibitor with an IC50 of 24 μM and a Ki of 0.6 μM. SMI-4a also inhibits Pim-2 (IC50 of 100 μM), and does not significantly inhibit the other serine/threonine- or tyrosine-kinases. SMI-4a has anticancer activity.
体外研究：
SMI-4a (0.5 μM；1 小时；HEK-293T 细胞) 处理会减弱完整细胞中标记的 Pim-1 的自身磷酸化。
产品资料
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