产品
编 号：F331862
分子式：C25H27N3O5S
分子量：481.56
分子式：C25H27N3O5S
分子量：481.56
产品类型
规格
价格
是否有货
5mg
询价
询价
结构图
CAS No: 350992-13-1
产品详情
生物活性：
Bifeprunox mesylate is a potent dopamine D2-like and 5-HT1A receptor partial agonist with pKis of 7.19 and 8.83 for cortex 5-HT1A and striatum D2, and a pEC50 of 6.37 for hippocampus 5-HT1A, respectively. Bifeprunox mesylate is an antipsychotic for the research of schizophrenia.
体内研究：
Bifeprunox (0.001-2.5 mg/kg) reduces marble burying in mice.Bifeprunox (4-250 μg/kg) influences nicotine-seeking behaviour in response to drug-associated stimuli in rats.
体外研究：
Bifeprunox has a pKi of 8 at h5-HT1A receptors, with an Emax of 70%.
Bifeprunox mesylate is a potent dopamine D2-like and 5-HT1A receptor partial agonist with pKis of 7.19 and 8.83 for cortex 5-HT1A and striatum D2, and a pEC50 of 6.37 for hippocampus 5-HT1A, respectively. Bifeprunox mesylate is an antipsychotic for the research of schizophrenia.
体内研究：
Bifeprunox (0.001-2.5 mg/kg) reduces marble burying in mice.Bifeprunox (4-250 μg/kg) influences nicotine-seeking behaviour in response to drug-associated stimuli in rats.
体外研究：
Bifeprunox has a pKi of 8 at h5-HT1A receptors, with an Emax of 70%.
产品资料
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