产品
编 号:F319424
分子式:C16H14O4
分子量:270.28
产品类型
结构图
CAS No: 32383-76-9
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产品详情
生物活性:
Medicarpin is a flavonoid isolated from Medicago sativa. Medicarpin induces apoptosis and overcome multidrug resistance in leukemia P388 cells by modulating P-gp-mediated efflux of agents.
体外研究:
Medicarpin (90 μM; for 48 h) triggers apoptosis in sensitive as well as multidrug resistant P388 cells. P-glycoprotein-expressing P388/DOX cells does not show resistance to medicarpin (IC50≈90 μM for P388 and P388/DOX cells).