产品
编 号:F281765
分子式:C22H28N4O3
分子量:396.48
产品类型
结构图
CAS No: 2247890-13-5
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产品详情
生物活性:
BAY-6035 is a potent, selective and substrate-competitive inhibitor of SMYD3. BAY-6035 inhibits methylation of MEKK2 peptide with an IC50 of 88 nM.
体外研究:
BAY-6035 inhibits in vitro methylation of MEKK2 peptide with an IC50 of 88 nM and has more than 100-fold selectivity over other histone methyltransferases. BAY-6035 inhibits the methylation of MEKK2 in cells with an IC50 of 70 nM.