产品
编 号:F280594
分子式:C41H41N9O8
分子量:787.82
产品类型
结构图
CAS No: 2231744-29-7
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产品详情
生物活性:
MT-802 is a potent BTK degrader based on Cereblon ligand, with a DC50 of 1 nM. MT-802 has potential to treat C481S mutant chronic lymphocytic leukemia (CLL).
体外研究:
MT-802 degrades BTK with a DC50 of 9.1 nM with maximal degradation being observed by 250 nM.