产品
编 号：F244118
分子式：C29H36N4O3
分子量：488.62
分子式：C29H36N4O3
分子量：488.62
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CAS No: 1962928-21-7
产品详情
生物活性：
PF-CBP1 is a highly selective inhibitor of the CREB binding protein bromodomain.
体外研究：
PF-CBP1 modulates key inflammatory genes in primary macrophages. PF-CBP1 downregulates RGS4 in neurons, a target linked to Parkinson's disease. PF-CBP1 is 139-fold selective over BRD4 in the biochemical assays and >105-fold selective by ITC.F-CBP1 is also a potent inhibitor of EP300 (a result observed for other CBP inhibitors.
PF-CBP1 is a highly selective inhibitor of the CREB binding protein bromodomain.
体外研究：
PF-CBP1 modulates key inflammatory genes in primary macrophages. PF-CBP1 downregulates RGS4 in neurons, a target linked to Parkinson's disease. PF-CBP1 is 139-fold selective over BRD4 in the biochemical assays and >105-fold selective by ITC.F-CBP1 is also a potent inhibitor of EP300 (a result observed for other CBP inhibitors.
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