产品
编 号:F238620
分子式:C6H13NO4
分子量:163.17
产品类型
结构图
CAS No: 19130-96-2
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生物活性:
1-Deoxynojirimycin (Duvoglustat) is a potent and orally active α-glucosidase inhibitor. 1-Deoxynojirimycin suppresses postprandial blood glucose and is widely used for diabetes mellitus. 1-Deoxynojirimycin possesses antihyperglycemic, anti-obesity, and antiviral features.
体内研究:
1-Deoxynojirimycin (Duvoglustat) (20 -80 mg/kg;iv;每日一次,持续 4 周) 显示抗肥胖作用。1-Deoxynojirimycin 通过激活显著改善胰岛素敏感性 db/db 小鼠骨骼肌胰岛素信号通路 PI3K/AKT。Animal Model:db/db mice
Dosage:20, 40, 80 mg/kg
Administration:Intravenously; daily for four weeks
Result:Significantly reduced body weight, blood glucose and serum insulin levels; Improved glucose tolerance and insulin tolerance.