产品
编 号:F238393
分子式:C22H27N5O3
分子量:409.48
产品类型
结构图
CAS No: 1910124-24-1
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产品详情
生物活性:
GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. GSK6853 shows excellent BRPF1 potency (pKd=9.5) and greater than 1600-fold selectivity over all other bromodomains.
体内研究:
The ip route of administration would be suitable for dosing GSK6853 in potential PK/PD models.