产品
编 号:F229151
分子式:C36H48N6O3
分子量:612.8
产品类型
结构图
CAS No: 1826865-46-6
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生物活性:
ZLD1039 is a potent, highly selective, and orally bioavailable EZH2 inhibitor. ZLD1039 shows potent and concentration-dependent inhibition of PRC2 enzymatic activity against EZH2 wild-type as well as Y641F, and A677G mutant enzymes with IC50 values of 5.6, 15, and 4.0?nM, respectively. ZLD1039 inhibits breast tumor growth and metastasis.