产品
编 号:F209356
分子式:C16H17ClNO5P
分子量:369.74
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10mM*1mL in DMSO
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5mg
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10mg
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50mg
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生物活性:
SDZ 220-581 is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7.

体内研究:
SDZ 220-581 (3.2-32 mg/kg; oral administration; for 24 hours; male OF-l mice) treatment dose-dependently protects mice against maximal electroshock seizures (MES). The time-course of protection by SDZ 220-581 is characterized by a rapid onset and long duration of action.Animal Model:Male OF-l mice (18-26 g)
Dosage:3.2 mg/kg, 10 mg/kg, 32 mg/kg
Administration:Oral administration; for 24 hours
Result:Dose-dependently protected mice against maximal electroshock seizures (MES) upon oral administration.
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