产品
编 号：F195853
分子式：C11H8F3N3O
分子量：255.2
分子式：C11H8F3N3O
分子量：255.2
产品类型
规格
价格
是否有货
10mM*1mL in DMSO
询价
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1mg
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5mg
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10mg
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25mg
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50mg
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结构图
CAS No: 1629633-48-2
产品详情
生物活性：
CDK8-IN-1 is a potent and selective CDK8 inhibitor with an IC50 of 3 nM.
体内研究：
CDK8-IN-1 displays low systemic clearance, very good exposure and oral bioavailability. The tmax is 0.25 h by PO. The mean values of Cmax are 9940 μg/L, 12740 μg/L by IV and PO respectively. The values of AUC are 9378, 25952 by IV and PO respectively.
CDK8-IN-1 is a potent and selective CDK8 inhibitor with an IC50 of 3 nM.
体内研究：
CDK8-IN-1 displays low systemic clearance, very good exposure and oral bioavailability. The tmax is 0.25 h by PO. The mean values of Cmax are 9940 μg/L, 12740 μg/L by IV and PO respectively. The values of AUC are 9378, 25952 by IV and PO respectively.
产品资料
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