产品
编 号:F194949
分子式:C30H35N3O3
分子量:485.62
产品类型
结构图
CAS No: 162408-66-4
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产品详情
生物活性:
GR 103691 is a potent, selective dopamine D3 receptor antagonist with a Ki value of 0.4 nM. GR 103691 shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites.
体外研究:
GR 103691 shows marked affinity for serotonin1A (5-HT1A) receptors (Ki of 5.8 nM) and α-1 adrenoceptors (Ki of 12.6 nM).