产品
编 号:F194526
分子式:C31H30ClN7O2
分子量:568.07
产品类型
结构图
CAS No: 1621523-07-6
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产品详情
生物活性:
THZ1-R is a non-cysteine reactive analog of THZ1 which displays diminished activity for CDK7 inhibition. THZ1-R binds to CDK7 with a Kd of 142 nM.
体外研究:
THZ1-R shows lower affinity at CDK7 than THZ1, with IC50 of 146 nM.